• 337 Citations
20012023
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  • 4 Similar Profiles
HIV Protease Inhibitors Medicine & Life Sciences
Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels Chemical Compounds
Protease Inhibitors Chemical Compounds
Neoplasms Medicine & Life Sciences
Scaffolds Chemical Compounds
Ligands Medicine & Life Sciences
Therapeutics Medicine & Life Sciences
Assays Chemical Compounds

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Grants 2011 2023

Neuropharmacology
Pharmaceutical Preparations
Ligands
Technology
Neurobiology
Kidney
Kidney Diseases
Research Personnel
Therapeutics
Nanomedicine
Antidepressive Agents
High-Throughput Screening Assays
Manuscripts
Organized Financing
Research
CXC Chemokines
MAP Kinase Signaling System
Chemokine Receptors
Chemokines
Prostatic Neoplasms
Astemizole
Castration
Nuclear Factor 90 Proteins
Prostatic Neoplasms
Zinc Compounds

Research Output 2001 2019

  • 337 Citations
  • 19 Article
  • 2 Review article
  • 1 Chapter

Discovery of a novel class of potent and selective tetrahydroindazole-based sigma-1 receptor ligands

Iyamu, I. D., Lv, W., Malik, N., Mishra, R. K. & Schiltz, G. E., May 1 2019, In : Bioorganic and Medicinal Chemistry. 27, 9, p. 1824-1835 12 p.

Research output: Contribution to journalArticle

Protein Transport
Ligands
Molecular modeling
Central Nervous System Diseases
Structure-Activity Relationship
Fluorine
Palladium
Bioactivity
Biological Products
Scaffolds

Regulation of MLL/COMPASS stability through its proteolytic cleavage by taspase1 as a possible approach for clinical therapy of leukemia

Zhao, Z., Wang, L., Volk, A. G., Birch, N. W., Stoltz, K. L., Bartom, E. T., Marshall, S. A., Rendleman, E. J., Nestler, C. M., Shilati, J., Schiltz, G. E., Crispino, J. D. & Shilatifard, A., Jan 1 2019, In : Genes and Development. 33, 1-2, p. 61-74 14 p.

Research output: Contribution to journalArticle

Aspartate Ammonia-Lyase
Threonine
Leukemia
Casein Kinase II
Therapeutics

Synthesis and Biological Evaluation of 3-Arylindazoles as Selective MEK4 Inhibitors

Deibler, K. K., Schiltz, G. E., Clutter, M., Mishra, R. K., Vagadia, P. P., O'Connor, M., George, M. D., Gordon, R., Fowler, G., Bergan, R. & Scheidt, K. A., Mar 22 2019, In : ChemMedChem. 14, 6, p. 615-620 6 p.

Research output: Contribution to journalArticle

MAP Kinase Kinase 4
Benzoic Acid
Molecular modeling
Oncology
p38 Mitogen-Activated Protein Kinases
1 Citation (Scopus)

Synthesis of a novel fused pyrrolodiazepine-based library with anti-cancer activity

Malik, N., Iyamu, I. D., Scheidt, K. A. & Schiltz, G. E., Apr 11 2018, In : Tetrahedron Letters. 59, 15, p. 1513-1516 4 p.

Research output: Contribution to journalArticle

Libraries
Succinimides
Scaffolds
Acylation
Neoplasms