Grants per year
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- 4 Similar Profiles
HIV Protease Inhibitors
Medicine & Life Sciences
Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels
Chemical Compounds
Protease Inhibitors
Chemical Compounds
Neoplasms
Medicine & Life Sciences
Scaffolds
Chemical Compounds
Ligands
Medicine & Life Sciences
Therapeutics
Medicine & Life Sciences
Assays
Chemical Compounds
Network
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Grants 2011 2023
DART2.0: comprehensive cell type-specific behavioral neuropharmacology
Duke University, National Institute of Mental Health
9/14/18 → 9/13/21
Project: Research project
Neuropharmacology
Pharmaceutical Preparations
Ligands
Technology
Neurobiology
Subproject for SP0046885 Luo Core B
Jin, J., Kandela, I., Luo, X., Mathew, J., Schiltz, G. E., Scott, E. A., Vanoye, C. G. & Wertheim, J. A.
National Institute of Diabetes, Digestive and Kidney Diseases
8/1/18 → 7/31/23
Project: Research project
Kidney
Kidney Diseases
Research Personnel
Therapeutics
Nanomedicine
Discovery of novel small molecule antidepressants
Clutter, M., Mishra, R. K. & Schiltz, G. E.
Vanderbilt University, National Institute of Mental Health
2/1/18 → 1/31/20
Project: Research project
Antidepressive Agents
High-Throughput Screening Assays
Manuscripts
Organized Financing
Research
Targeting chemokine signaling and MAPK/ERK pathway in advanced prostate cancer
Yu, J., Cristofanilli, M., Hussain, M., Miller, R. J., Schiltz, G. E., Yang, X. J., Zhang, B. & Zhao, C.
12/31/17 → 12/31/19
Project: Research project
CXC Chemokines
MAP Kinase Signaling System
Chemokine Receptors
Chemokines
Prostatic Neoplasms
Targeting EZH2 in castration-resistant prostate cancer
Mishra, R. K. & Schiltz, G. E.
U.S. Army Medical Research and Materiel Command
8/1/17 → 7/31/20
Project: Research project
Astemizole
Castration
Nuclear Factor 90 Proteins
Prostatic Neoplasms
Zinc Compounds
Research Output 2001 2019
Discovery of a novel class of potent and selective tetrahydroindazole-based sigma-1 receptor ligands
Iyamu, I. D., Lv, W., Malik, N., Mishra, R. K. & Schiltz, G. E., May 1 2019, In : Bioorganic and Medicinal Chemistry. 27, 9, p. 1824-1835 12 p.Research output: Contribution to journal › Article
Protein Transport
Ligands
Molecular modeling
Central Nervous System Diseases
Structure-Activity Relationship
Palladium-Catalyzed Coupling Reactions on Functionalized 2-Trifluoromethyl-4-chromenone Scaffolds: Synthesis of Highly Functionalized Trifluoromethyl Heterocycles
Izquierdo, J., Jain, A. D., Abdulkadir, S. A. & Schiltz, G. E., Jan 1 2019, In : Synthesis (Germany). 51, 6, p. 1342-1352 11 p.Research output: Contribution to journal › Article
Fluorine
Palladium
Bioactivity
Biological Products
Scaffolds
Regulation of MLL/COMPASS stability through its proteolytic cleavage by taspase1 as a possible approach for clinical therapy of leukemia
Zhao, Z., Wang, L., Volk, A. G., Birch, N. W., Stoltz, K. L., Bartom, E. T., Marshall, S. A., Rendleman, E. J., Nestler, C. M., Shilati, J., Schiltz, G. E., Crispino, J. D. & Shilatifard, A., Jan 1 2019, In : Genes and Development. 33, 1-2, p. 61-74 14 p.Research output: Contribution to journal › Article
Aspartate Ammonia-Lyase
Threonine
Leukemia
Casein Kinase II
Therapeutics
Synthesis and Biological Evaluation of 3-Arylindazoles as Selective MEK4 Inhibitors
Deibler, K. K., Schiltz, G. E., Clutter, M., Mishra, R. K., Vagadia, P. P., O'Connor, M., George, M. D., Gordon, R., Fowler, G., Bergan, R. & Scheidt, K. A., Mar 22 2019, In : ChemMedChem. 14, 6, p. 615-620 6 p.Research output: Contribution to journal › Article
MAP Kinase Kinase 4
Benzoic Acid
Molecular modeling
Oncology
p38 Mitogen-Activated Protein Kinases
1
Citation
(Scopus)
Synthesis of a novel fused pyrrolodiazepine-based library with anti-cancer activity
Malik, N., Iyamu, I. D., Scheidt, K. A. & Schiltz, G. E., Apr 11 2018, In : Tetrahedron Letters. 59, 15, p. 1513-1516 4 p.Research output: Contribution to journal › Article
Libraries
Succinimides
Scaffolds
Acylation
Neoplasms