Datasets
- 18 results
Search results
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Additional file 2: Table S2. of Retention of normal glia function by an isoform-selective protein kinase inhibitor drug candidate that modulates cytokine production and cognitive outcomes
Zhou, Z. (Contributor), Bachstetter, A. D. (Creator), Späni, C. B. (Creator), Roy, S. M. (Contributor), Watterson, D. M. (Contributor) & Van Eldik, L. J. (Contributor), figshare, 2017
DOI: 10.6084/m9.figshare.c.3735430_d2.v1, https://springernature.figshare.com/articles/dataset/Additional_file_2_Table_S2_of_Retention_of_normal_glia_function_by_an_isoform-selective_protein_kinase_inhibitor_drug_candidate_that_modulates_cytokine_production_and_cognitive_outcomes/4822510/1
Dataset
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4YPD : Crystal Structure of DAPK1 catalytic domain in complex with the hinge binding fragment 4-methylpyridazine
Watterson, D. M. (Contributor), Grum-Tokars, V. (Contributor), Roy, S. M. (Contributor), Minasov, G. (Contributor) & Anderson, W. F. (Contributor), RCSB-PDB, 2015
DOI: 10.2210/pdb4ypd/pdb, https://www.rcsb.org/structure/4YPD
Dataset
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CCDC 1851508: Experimental Crystal Structure Determination
Roy, S. M. (Contributor), Watterson, D. M. (Contributor) & Malliakas, C. (Contributor), Cambridge Crystallographic Data Centre, 2018
DOI: 10.5517/ccdc.csd.cc204n2x, http://www.ccdc.cam.ac.uk/services/structure_request?id=doi:10.5517/ccdc.csd.cc204n2x&sid=DataCite
Dataset
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Human P38alpha MAPK in Complex with a Novel and Selective Small Molecule Inhibitor
Watterson, D. M. (Contributor), Grum-Tokars, V. L. (Contributor), Roy, S. M. (Contributor), Schavocky, J. P. (Contributor), de Bradaric, B. (Contributor), Bachstetter, A. D. (Contributor), Xing, B. (Contributor), Dimayuga, E. (Contributor), Saeed, F. (Contributor), Zhang, H. (Contributor), Staniszewski, A. (Contributor), Pelletier, J. C. (Contributor), Minasov, G. (Contributor), Anderson, W. F. (Contributor), Arancio, O. (Contributor) & van Eldik, L. J. (Contributor), Protein Data Bank (PDB), Jun 5 2013
DOI: 10.2210/pdb4F9W/pdb, https://www.wwpdb.org/pdb?id=pdb_00004f9w
Dataset
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Structure of human p38aMAPK-arylpyridazinylpyridine fragment complex used in inhibitor discovery
Roy, S. M. (Contributor), Minasov, G. (Contributor), Arancio, O. (Contributor), Chico, L. W. (Contributor), Van Eldik, L. J. (Contributor), Anderson, W. F. (Contributor), Pelletier, J. C. (Contributor) & Watterson, D. M. (Contributor), Protein Data Bank (PDB), Jun 22 2016
DOI: 10.2210/pdb4ZTH/pdb, https://www.wwpdb.org/pdb?id=pdb_00004zth
Dataset
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Human p38 alpha MAPK in complex with a pyridazine based inhibitor
Munoz, L. (Contributor), Ranaivo, H. (Contributor), Roy, S. M. (Contributor), Hu, W. (Contributor), Craft, J. M. (Contributor), McNamara, L. K. (Contributor), Chico, L. W. (Contributor), Van Eldik, L. J. (Contributor), Watterson, D. M. (Contributor), Minasov, G. (Contributor), Arancio, O. (Contributor), Anderson, W. F. (Contributor) & Pelletier, J. C. (Contributor), Protein Data Bank (PDB), Jun 27 2012
DOI: 10.2210/pdb4EWQ/pdb, https://www.wwpdb.org/pdb?id=pdb_00004ewq
Dataset
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Crystal structure of p38 alpha MAP kinase in complex with a novel isoform selective drug candidate
Roy, S. M. (Contributor), Grum-Tokars, V. L. (Contributor), Schavocky, J. P. (Contributor), Saeed, F. (Contributor), Staniszewski, A. (Contributor), Teich, A. F. (Contributor), Arancio, O. (Contributor), Bachstetter, A. D. (Contributor), Webster, S. J. (Contributor), Van Eldik, L. J. (Contributor), Minasov, G. (Contributor), Anderson, W. F. (Contributor), Pelletier, J. C. (Contributor) & Watterson, D. M. (Contributor), Protein Data Bank (PDB), Feb 25 2015
DOI: 10.2210/pdb4R3C/pdb, https://www.wwpdb.org/pdb?id=pdb_00004r3c
Dataset
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Human P38 alpha MAPK In Complex With a Novel and Selective Small Molecule Inhibitor
Watterson, D. M. (Contributor), Grum-Tokars, V. L. (Contributor), Roy, S. M. (Contributor), Schavocky, J. P. (Contributor), de Bradaric, B. (Contributor), Bachstetter, A. D. (Contributor), Xing, B. (Contributor), Dimayuga, E. (Contributor), Saeed, F. (Contributor), Zhang, H. (Contributor), Staniszewski, A. (Contributor), Pelletier, J. C. (Contributor), Minasov, G. (Contributor), Anderson, W. F. (Contributor), Arancio, O. (Contributor) & van Eldik, L. J. (Contributor), Protein Data Bank (PDB), Jun 5 2013
DOI: 10.2210/pdb4F9Y/pdb, https://www.wwpdb.org/pdb?id=pdb_00004f9y
Dataset
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Retention of normal glia function by an isoform-selective protein kinase inhibitor drug candidate that modulates cytokine production and cognitive outcomes
Zhou, Z. (Contributor), Bachstetter, A. D. (Creator), Späni, C. B. (Creator), Roy, S. M. (Contributor), Watterson, D. M. (Contributor) & Van Eldik, L. J. (Contributor), figshare, 2017
DOI: 10.6084/m9.figshare.c.3735430.v1, https://figshare.com/collections/Retention_of_normal_glia_function_by_an_isoform-selective_protein_kinase_inhibitor_drug_candidate_that_modulates_cytokine_production_and_cognitive_outcomes/3735430/1
Dataset
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Additional file 1: Table S1. of Retention of normal glia function by an isoform-selective protein kinase inhibitor drug candidate that modulates cytokine production and cognitive outcomes
Zhou, Z. (Contributor), Bachstetter, A. D. (Creator), Späni, C. B. (Creator), Roy, S. M. (Contributor), Watterson, D. M. (Contributor) & Van Eldik, L. J. (Contributor), figshare, 2017
DOI: 10.6084/m9.figshare.c.3735430_d1, https://springernature.figshare.com/articles/dataset/Additional_file_1_Table_S1_of_Retention_of_normal_glia_function_by_an_isoform-selective_protein_kinase_inhibitor_drug_candidate_that_modulates_cytokine_production_and_cognitive_outcomes/4822489
Dataset
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Additional file 4: Table S4. of Retention of normal glia function by an isoform-selective protein kinase inhibitor drug candidate that modulates cytokine production and cognitive outcomes
Zhou, Z. (Contributor), Bachstetter, A. D. (Creator), Späni, C. B. (Creator), Roy, S. M. (Contributor), Watterson, D. M. (Contributor) & Van Eldik, L. J. (Contributor), figshare, 2017
DOI: 10.6084/m9.figshare.c.3735430_d4.v1, https://springernature.figshare.com/articles/dataset/Additional_file_4_Table_S4_of_Retention_of_normal_glia_function_by_an_isoform-selective_protein_kinase_inhibitor_drug_candidate_that_modulates_cytokine_production_and_cognitive_outcomes/4822558/1
Dataset
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4R3C : Crystal structure of p38 alpha MAP kinase in complex with a novel isoform selective drug candidate
Roy, S. M. (Contributor), Grum-Tokars, V. L. (Contributor), Minasov, G. (Contributor), Anderson, W. F. (Contributor) & Watterson, D. M. (Contributor), RCSB-PDB, 2015
DOI: 10.2210/pdb4r3c/pdb, https://www.rcsb.org/structure/4R3C
Dataset
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Crystal Structure of DAPK1 catalytic domain in complex with the hinge binding fragment 4-methylpyridazine
McNamara, L. K. (Contributor), Brunzelle, J. S. (Contributor), Schavocky, J. P. (Contributor), Watterson, D. M. (Contributor), Grum-Tokars, V. (Contributor), Roy, S. M. (Contributor), de Bradaric, B. (Contributor), Bachstetter, A. D. (Contributor), Xing, B. (Contributor), Dimayuga, E. (Contributor), Saeed, F. (Contributor), Zhang, H. (Contributor), Staniszewski, A. (Contributor), Pelletier, J. C. (Contributor), Minasov, G. (Contributor), Anderson, W. F. (Contributor), Arancio, O. (Contributor) & van Eldik, L. J. (Contributor), Protein Data Bank (PDB), May 13 2015
DOI: 10.2210/pdb4YPD/pdb, https://www.wwpdb.org/pdb?id=pdb_00004ypd
Dataset
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4YO4 : Crystal Structure of DAPK1 catalytic domain in complex with the hinge binding fragment phthalazine
Watterson, D. M. (Contributor), Grum-Tokars, V. L. (Contributor), Roy, S. M. (Contributor), Minasov, G. (Contributor) & Anderson, W. F. (Contributor), RCSB-PDB, 2015
DOI: 10.2210/pdb4yo4/pdb, https://www.rcsb.org/structure/4YO4
Dataset
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Human P38 alpha Mitogen-Activated Kinase In Complex With SB239063
Watterson, D. M. (Contributor), Grum-Tokars, V. L. (Contributor), Roy, S. M. (Contributor), Schavocky, J. P. (Contributor), de Bradaric, B. (Contributor), Bachstetter, A. D. (Contributor), Xing, B. (Contributor), Dimayuga, E. (Contributor), Saeed, F. (Contributor), Zhang, H. (Contributor), Staniszewski, A. (Contributor), Pelletier, J. C. (Contributor), Minasov, G. (Contributor), Anderson, W. F. (Contributor), Arancio, O. (Contributor) & van Eldik, L. J. (Contributor), Protein Data Bank (PDB), Jun 5 2013
DOI: 10.2210/pdb4FA2/pdb, https://www.wwpdb.org/pdb?id=pdb_00004fa2
Dataset
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CCDC 1851509: Experimental Crystal Structure Determination
Roy, S. M. (Contributor), Watterson, D. M. (Contributor) & Malliakas, C. (Contributor), Cambridge Crystallographic Data Centre, 2018
DOI: 10.5517/ccdc.csd.cc204n3y, http://www.ccdc.cam.ac.uk/services/structure_request?id=doi:10.5517/ccdc.csd.cc204n3y&sid=DataCite
Dataset
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Additional file 3: Table S3. of Retention of normal glia function by an isoform-selective protein kinase inhibitor drug candidate that modulates cytokine production and cognitive outcomes
Zhou, Z. (Contributor), Bachstetter, A. D. (Creator), Späni, C. B. (Creator), Roy, S. M. (Contributor), Watterson, D. M. (Contributor) & Van Eldik, L. J. (Contributor), figshare, 2017
DOI: 10.6084/m9.figshare.c.3735430_d3.v1, https://springernature.figshare.com/articles/dataset/Additional_file_3_Table_S3_of_Retention_of_normal_glia_function_by_an_isoform-selective_protein_kinase_inhibitor_drug_candidate_that_modulates_cytokine_production_and_cognitive_outcomes/4822528/1
Dataset
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4EWQ : Human p38 alpha MAPK in complex with a pyridazine based inhibitor
Roy, S. M. (Contributor), Watterson, D. M. (Contributor), Grum-Tokars, V. L. (Contributor), Schavocky, J. P. (Contributor), Minasov, G. (Contributor) & Anderson, W. F. (Contributor), RCSB-PDB, 2012
DOI: 10.2210/pdb4ewq/pdb, https://www.rcsb.org/structure/4EWQ
Dataset