Abstract
1,2,3-Triazoles were prepared in good to modest yields by cycloaddition of alkyl azides onto enol ethers under solventless conditions. The reaction can access ring-fused triazoles that are unavailable by azide-alkyne cycloadditions and is easily scalable. The 1,2,3-triazole products bear functionality that may be readily derivatized.
Original language | English (US) |
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Article number | M10204SS |
Pages (from-to) | 2497-2502 |
Number of pages | 6 |
Journal | Synthesis |
Issue number | 15 |
DOIs | |
State | Published - Oct 4 2005 |
Externally published | Yes |
Keywords
- Azides
- Cycloadditions
- Heterocycles
- Nitrogen
- Regioselectivity
ASJC Scopus subject areas
- Catalysis
- Organic Chemistry