Validation of Human Sterol 14α-Demethylase (CYP51) Druggability: Structure-Guided Design, Synthesis, and Evaluation of Stoichiometric, Functionally Irreversible Inhibitors

Laura Friggeri, Tatiana Y. Hargrove, Zdzislaw Wawrzak, F. Peter Guengerich, Galina I. Lepesheva*

*Corresponding author for this work

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